Lwm lub npe: androgen antagonists, androgen receptor blockers, testosterone blockers
Antiandrogens yog dab tsi?
Antiandrogens yog lub npe muab rau ntau pawg ntawm cov tshuaj uas tawm tsam qhov cuam tshuam ntawm cov txiv neej cov tshuaj hormones, testosterone thiab dihydrotestosterone. Txiv neej cov tshuaj hormones tseem hu ua androgens; antiandrogens kuj tseem hu ua androgen receptor blockers.
Qee cov antiandrogens ua haujlwm los ntawm kev txo qis lub cev tsim cov androgens thaum lwm tus thaiv androgen receptors, txwv lub cev lub peev xwm los siv cov androgens tsim.
Antiandrogens yog siv nyob rau hauv kev kho mob ntawm ntau yam mob thiab mob xws li mob qog noj ntshav prostate , precocious puberty hauv cov txiv neej hluas, benign prostatic hyperplasia , androgenic alopecia (txiv neej-pattern plaub hau poob ) thiab kev sib deev , xws li hyper-sexuality, hauv cov txiv neej.
Hauv cov poj niam, cov tshuaj antiandrogens tuaj yeem siv los kho cov mob polycystic zes qe menyuam, hirsutism (ntau lub ntsej muag lossis lub cev plaub hau), amenorrhea (tsis muaj kev coj khaub ncaws), pob txuv , thiab ob peb lwm yam mob.
Cov npe ntawm Antiandrogens:
Saib los ntawm Hom | Ntau Lim los ntawmTxhua yam mob Hirsutism Prostate CancerAvg. Kev ntsuas | Kev tshuaj xyuas | |
---|---|---|
Xtandi ( Pro ) Lub npe dav: enzalutamide | 4.5 | 12 kev tshuaj xyuas |
Casodex ( Pro ) Lub npe dav: tshuaj bicalutamide | 7.2 | 7 kev tshuaj xyuas |
yuam kev ( Pro ) Lub npe dav: apalutamide | 8.0 ib | 2 kev tshuaj xyuas |
Nubqa ( Pro ) Lub npe dav: darolutamide | tsis muaj kev tshuaj xyuas | |
Nilandron ( Pro ) Lub npe dav: nilutamide | tsis muaj kev tshuaj xyuas | |
Eulexin ( Pro ) Lub npe dav: flutamide | tsis muaj kev tshuaj xyuas | |
Rau kev ntsuam xyuas, cov neeg siv tau nug seb lawv pom cov tshuaj zoo npaum li cas thaum xav txog qhov zoo / qhov tsis zoo thiab kev siv yooj yim (1 = tsis zoo, 10 = zoo tshaj plaws). |
Cov ntaub ntawv ntxiv
Nco ntsoov sab laj nrog koj tus kws kho mob kom paub tseeb tias cov ntaub ntawv uas tshwm sim hauv nplooj ntawv no siv tau rau koj tus kheej.